Lewis acid-catalyzed hetero Diels-Alder cycloadditions of 3-alkyl, 3-phenyl and 3-carboxylated 2H-azirines
2001 (English)In: Tetrahedron Letters, ISSN 0040-4039, E-ISSN 1873-3581, Vol. 42, no 52, 9289-9291 p.Article in journal (Refereed) Published
Activation by Lewis acids of 3-alkyl and 3-phenyl 2H-azirines promotes their participation in hetero Diels-Alder reactions with a variety of dienes. This methodology circumvents the previous requirement of an electron-withdrawing carboxyl moiety at the 3-position of the 2H-azirine.
Place, publisher, year, edition, pages
2001. Vol. 42, no 52, 9289-9291 p.
chiral aziridines, dienophiles
IdentifiersURN: urn:nbn:se:kth:diva-21165ISI: 000172658200047OAI: oai:DiVA.org:kth-21165DiVA: diva2:339862
QC 201005252010-08-102010-08-10Bibliographically approved